Publications 2009

1. Saczewski, J.; Paluchowska, A.; Klenc, J.; Raux, E.; Barnes, S.; Sullivan, S.; Duszyńska, B.; Bojarski, A. J.; Strekowski, L. Synthesis of 4-substituted 2-(4-methylpiperazino)pyrimidines and quinazoline analogs as serotonin 5-HT2A receptor ligands. J. Heterocyclic Chem. 2009, 46, 1259-1265 (http://onlinelibrary.wiley.com/doi/10.1002/jhet.236/abstract).
2. Herold, F.; Izbicki, L.; Chodkowski, A.; Dawidowski, M.; Krol, M.; Kleps, J.; Turlo, J.; Wolska, I.; Nowak, G.; Stachowicz, K.; Dybala, M.; Siwek, A.; Nowak, M.; Pieniazek, E.; Jaronczyk, M.; Sylte, I.; Mazurek, A. P.  Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT1A activity: part 2. Eur. J. Med. Chem. 2009, 44, 4702-4715
(http://www.ncbi.nlm.nih.gov/pubmed/19665823)
3. Tokarski, K.; Pitra, P.; Duszynska, B.; Hess, G. Imipramine counteracts corticosterone-induced alterations in the effects of the activation of 5-HT(7) receptors in rat hippocampus. J. Physiol Pharmacol. 2009, 60, 83-88 (http://www.ncbi.nlm.nih.gov/pubmed/19617650).
4. Testa, B.; Vistoli, G.; Pedretti, A.; Bojarski, A. J. Atomic diversity, molecular diversity, and chemical diversity: the concept of chemodiversity. Chem. Biodivers. 2009, 6, 1145-1151 (http://www.ncbi.nlm.nih.gov/pubmed/19697332).
5. Zajdel, P.; Subra, G. ; Verdie, P.; Gabzdyl, E.; Bojarski, A. J.; Duszynska, B.; Martinez, J.; Pawlowski, M. Sulfonamides with the N-alkyl-N’-dialkylguanidine moiety as 5-HT7 receptor ligands. Bioorg. Med. Chem. Lett. 2009, 19, 4827-4831  (http://www.ncbi.nlm.nih.gov/pubmed/19560916).
6. Testa, B.; Bojarski, A. J. Simulations in evolution. II. Relative fitness and the propagation of mutants. Chem. Biodivers. 2009, 6, 356-368  (http://www.ncbi.nlm.nih.gov/pubmed/19319872). 
7. Badarau, E.; Suzenet, F.; Bojarski, A. J.; Finaru, A. L.; Guillaumet, G. Benzimidazolone-based serotonin 5-HT(1A) or 5-HT(7)R ligands: Synthesis and biological evaluation. Bioorg. Med. Chem. Lett. 2009, 19, 1600-1603 (http://www.ncbi.nlm.nih.gov/pubmed/19237285).
8. Bojarski, A. J.; Kuran, B.; Kossakowski, J.; Koziol, A. ; Jagiello-Wojtowicz, E.; Chodkowska, A. Synthesis and serotonin receptor activity of the arylpiperazine alkyl/propoxy derivatives of new azatricycloundecanes. Eur. J. Med. Chem. 2009, 44, 152-164  (http://www.ncbi.nlm.nih.gov/pubmed/18486277).
9. Zajdel, P.; Subra, G. ; Verdie, P.; Bojarski, A. J.; Duszynska, B.; Basista, K.; Obniska, J.; Martinez, J.; Pawlowski, M. The influence of an ethylene spacer on the 5-HT(1A) and 5-HT(2A) receptor affinity of arylpiperazine derivatives of amides with N-acylated amino acids and 3-differently substituted pyrrolidine-2,5-diones. Eur. J. Med. Chem. 2009, 44, 800-808 (http://www.ncbi.nlm.nih.gov/pubmed/18603331).