Publications 2017

  1. Satała, G.; Duszyńska, B.; Lenda, T.; Nowak, G.; Bojarski, A.J. Allosteric Inhibition of Serotonin 5-HT7 Receptors by Zinc Ions. Mol Neurobiol. 2017 [Epub ahead of print] (https://www.ncbi.nlm.nih.gov/pubmed/28455702)
  2. Hogendorf, A.S.; Hogendorf, A.; Kurczab, R.; Satała, G.; Lenda, T.; Walczak, M.; Latacz, G.; Handzlik, J.; Kieć-Kononowicz, K.; Wierońska, J.M.; Woźniak, M.; Cieślik, P.; Bugno, R.; Staroń, J.; Bojarski, A.J. Low-basicity 5-HT7 Receptor Agonists Synthesized Using the van Leusen Multicomponent Protocol. Sci Rep. 2017 7, 1444 (https://www.ncbi.nlm.nih.gov/pubmed/28473721)
  3. Partyka, A.; Kurczab, R.; Canale, V.; Satała, G.; Marciniec, K.; Pasierb, A.; Jastrzębska-Więsek, M.; Pawłowski, M.; Wesołowska, A.; Bojarski, A.J.; Zajdel, P. The impact of the halogen bonding on D2 and 5-HT1A/5-HT7 receptor activity of azinesulfonamides of 4-[(2-ethyl)piperidinyl-1-yl]phenylpiperazines with antipsychotic and antidepressant properties. Bioorg Med Chem. 2017 25, 3638-3648 (https://www.ncbi.nlm.nih.gov/pubmed/28529043)
  4. Intagliata, S.; Modica, M. N.; Pittalà, V.; Salerno, L.; Siracusa, M. A.; Cagnotto, A.; Salmona, M.; Kurczab, R.; Romeo, G. New N- and O-arylpiperazinylalkyl pyrimidines and 2-methylquinazolines derivatives as 5-HT7 and 5-HT1A receptor ligands: Synthesis, structure-activity relationships, and molecular modeling studies. Bioorg. Med. Chem. 2017, 25, 1250–1259 (https://www.ncbi.nlm.nih.gov/pubmed/28063784)
  5. Warszycki, D.; Rueda, M.;, Mordalski, S.; Kristiansen, K.; Satała, G.; Rataj, K.; Chilmonczyk, Z.; Sylte, I.; Abagyan, R.; Bojarski, A. J. From Homology Models to a Set of Predictive Binding Pockets-a 5-HT1A Receptor Case Study. J Chem Inf Model. 2017 [Epub ahead of print] (https://www.ncbi.nlm.nih.gov/pubmed/28055203)
  6. Leśniak, D.; Jastrzębski, S.; Podlewska, S.; Czarnecki, W. M.; Bojarski, A. J. Quo vadis G protein-coupled receptor ligands? A tool for analysis of the emergence of new groups of compounds over time. Bioorg Med Chem Lett. 2017, 27, 626-631 (https://www.ncbi.nlm.nih.gov/pubmed/27993519).
  7. Hogendorf, A. S.; Hogendorf, A.; Kurczab, R.; Satała, G.; Lenda, T.; Walczak, M.; Latacz, G.; Handzlik, J.; Kieć-Kononowicz, K.; Wierońska, J.; Woźniak, M.; Cieślik, P.; Bugno, R.; Staroń, J.; Bojarski, A. J. Low-basicity 5-HT7 Receptor Agonists Synthesized Using the van Leusen Multicomponent Protocol Sci. Rep. 2017, 7, Article number: 1444 (http://www.nature.com/articles/s41598-017-00822-4).
  8. Staroń, J.; Mordalski, S.; Warszycki, D.; Satała, G.; Hogendorf, A. S.; Bojarski, A. J. Pyrano[2,3,4-cd]indole as a Scaffold for Selective Nonbasic 5-HT6R Ligands ACS Med. Chem. Lett. 2017, 8(4), pp 390–394