Conferences 2011

1. The 47th Norwegian Biochemical Society (NBS) contact meeting, 03-06.02.2011, Norway

  • Gabrielsen, M.; Kurczab, R.; Jarończyk, M.; Ravna, A.W.; Kristiansen, K.; Chilmonczyk, Z.; Bojarski, A.J.; Sylte, I.; Docking of substrates and inhibitors into the substrate binding site of two serotonin transporter models; Book of Abstracts, p.39.Abstract
  • Kristiansen, K.; Rueada, M.; Warszycki, D.; Kurczab, R.; Gabrielsen, M.; Abagyan, R.; Bojarski, A.J.; Sylte, I.; Modeling of ligand interactions for the human 5-HT1A receptor. Docking, pharmacophores and virtual screening of databases containing drug-like compounds; Book of Abstracts, p.108. Abstract

2. Spring Congress of Polish Chemical Society Student Section, 13-17.04.2011, Murzasichle, Poland

  •  Smusz, S.; Kurczab, R.; Warszycki, D.; Kościółek, T.; Mordalski, S.; Bojarski, A.J.; Hybridization of ligands as a way of generating combinatorial libraries of drug candidates; Book of Abstracts, p.130. Abstract Poster

3.  29th Informal Meeting on Mass Spectrometry, 18-19.05.2011, Primiero, Italy

  • Chilmonczyk, Z.; Kossakowski, J.; Nowak, G.; Bojarski, A.J.; Wołosewicz, K.; Gabrielsen, M.; Sylte, I.; Witowska-Jarosz, J.; New serotonin transporter inhibitors with antidepressant activity in mice by MS; Book of Abstracts, p.118.Abstract
  • Witowska-Jarosz, J.; Kossakowski, J.; Nowak, G.; Bojarski, A.J.; Wołosewicz, K.; Gabrielsen, M.; Sylte, I.; Baran, P.; Chilmonczyk, Z.; Mass spectrometry of new 6-nitroquipazine derivatives; Book of Abstracts, p.W6.Abstract

4. The Twentieth Days of Neuropsychopharmacology, 22-25.05.2011, Ustroń-Jaszowiec,Poland

  • Chilmonczyk, Z.; Kossakowski, J.; Walory, J.; Koronkiewicz, M.; Sylte, I.; Nowak, G.; Bojarski, A.J.; Influence of new high affinity serotonin transporter ligands on cellular cAMP levels; Pharmacological Reports, 2011, 63, p.565.
  • Brański, P.; Staroń, J.; Bugno, R.; Wierońska, J.; Bojarski, A.J.; Burnat, G.; Pałucha-Poniewiara, A.; Pilc, A.; Synthesis and characterization of novel metabotropic glutamate receptor 2/3 (mGluR2/3) positive allosteric modulator (PAM); Pharmacological Reports, 2011, 63, p.577.
  • Kościółek, T.; Mordalski, S.; Bojarski, A.J.; Different approaches in homology modeling of transmembrane domain of metabotropic glutamate receptor type 4 (mGluR4); Pharmacological Reports, 2011, 63, p.579. Abstract
  • Kurczab, R.; Bojarski, A.J.; How to find a needle in a haystack? The application of  in silico methods in searching of potentially new PAM of mGluR III; Pharmacological Reports, 2011, 63, p.579. Abstract

5. 9th International Conference on Chemical Structures, 05-09.06.2011, Noordwijkerhout, The Netherlands

  • Kurczab, R.; Bojarski, A.J.; The Multi-Conformations-Receptor-Based Pharmacophore Model Generation Schema and Its Potential Applications in Virtual Screening; Book of Abstracts, p.126. Abstract Poster
  • Warszycki, D.; Kristiansen, K.; Mordalski, S.; Kurczab, R.; Sylte, I.; Bojarski, A.J.; Comparison of various strategies in pharmacophore models generation – application to 5-HT1A receptor ligands; Book of Abstracts, p.95. Abstract Poster

6. VII Joint Meeting on Medicinal Chemistry, 26-27.06.2011, Catania, Italy

  • Chilmonczyk, Z.; Kossakowski, J.; Sylte, I.; Bojarski, A.J.; Nowak, G.; Wołosewicz, K.; New derivatives of nitroquipazine as potential antidepressive drugs; Book of Abstracts, p.167.Abstract
  • Kurczab, R.; Mordalski, S.; Kościółek, T.; Bojarski, A.J.; The new strategy in structure-based pharmacophore model generation and its applications in virtual screening; Book of Abstracts, p.187. Abstract Poster
  • Bugno, R.; Duszyńska, B.; Satała, G.; Mordalski, S.; Chmielarz, P.; Nalepa, I.; Bojarski, A.J.; Searching of novel leads for 5-HT7 receptor antagonists – selectivity hints from molecular modeling studies; Book of Abstracts, p.189. Abstract Poster
  • Warszycki, D.; Kristiansen, K.; Kurczab, R.; Satała, G.; Mordalski, S.; Sylte, I.; Bojarski, A.J.; Extensive pharmacophore modeling studies on 5-HT1A receptor ligands – single hypothesis vs. linear combinations; Book of Abstracts, p.186. Abstract Poster
  • Zajdel, P.; Marciniec, K.; Maślankiewicz, A.; Grychowska, K.; Satała, G.; Partyka, A.; Jastrzębska-Więsek, M.; Wróbel, D.; Wesolowska, A.; Bojarski, A.J.; Pawłowski, M.; Novel 5-HT7 receptor ligands N-terminated with quinolinesulfoamoyl moieties; Book of Abstracts, p.200. Abstract

7. 47th International Conference on Medicinal Chemistry, 06-08.07.2011, Lyon, France

  • Sagnes, C.; Fournet, G.; Satała, G.; Bojarski, A.J.; Joseph, B.; New N-arylindoles based serotonin 5-HT7 ligands: Synthesis and binding affinity studies; Book of Abstracts, p.P051.

8. 4th International Symposium on Advances in Synthetic and Medicinal Chemistry, 21-25.08.2011, St. Petersburg, Russia

  • Trela, M.; Bugno, R.; Kurczab, R.; Brański, P.; Bojarski, A.J.; New heterocyclic derivatives as potential allosteric modulators of group III metabotropic glutamate receptors; Book of Abstracts, p.220. Abstract Poster
  • Staroń, J.; Warszycki, D.; Satała, G.; Bugno, R.; Bojarski, A.J.; Bioisosterism, the use in designing 5-HT6 receptor ligands; Book of Abstracts, p.176. Abstract Poster
  • Stankiewicz, A.; Bugno, R.; Brański, P.; Bojarski, A.J.; 1,2,4-Oxadiazole derivatives as potential allosteric modulators of the mglur4; Book of Abstracts.Poster
  • Brański, P.; Staroń, J.; Bugno, R.; Wierońska, J.; Bojarski, A.; Burnat, G.; Chorobik, P.; Chruścicka, B.; Pałucha-Poniewiara, A.; Sławińska, A.; Stachowicz, K.; Pilc, A.; Discovery of novel and systemically active allosteric ligand of metabotropic glutamate receptor group II with potential anxiolytic properties; Book of Abstracts.

9. The 4th Conversatory of Medicinal Chemistry, 08-10.09.2011, Lublin, Poland

  • Witowska-Jarosz, J.; Kossakowski, J.; Nowak, G.; Bojarski, A.J.; Wołosewicz, K.; Gabrielsen, M.; Sylte, I.; Baran, P.; Mazurek, A.P.; Chilmonczyk, Z.; Mass Spectrometry of New Serotonin Transporter Inhibitors; Book of Abstracts, p.K-8.Abstract
  • Warszycki, D.; Kristiansen, K.; Kurczab, R.; Mordalski, S.; Sylte, I.; Bojarski, A.J.; Linear Combination of Pharmacophore Hypotheses as a New Tool in Search of New 5-HT1A Receptor Ligands; Book of Abstracts, p.PP-4. Abstract Poster
  • Dela, A.; Wójcik, R.; Duszyńska, B.; Satała, G.; Handzlik, J.; Bojarski, A.J.; Kieć-Kononowicz, K.; Influence of the Substituent(s) at Aromatic Rings at Arylidene Phenylpiperazine Hydantoin on Affinity to 5-HT6 and 5-HT7 Serotonine Receptors; Book of Abstracts, p.P-8.Abstract
  • Jarończyk, M.; Wołosewicz, K.; Nowak, G.; Gabrielsen, M.; Mazurek, A.P.; Ravna, A.W.; Bojarski, A.J.; Sylte, I.; Chilmonczyk, Z.; The study of buspirone analogues docking to serotonin transporter; Book of Abstracts, p.P-13. Abstract
  • Kurczab, R.; Zajdel, P.; Pawłowski, M.; Bojarski, A.J.; Development and Validation of Methodology for Designing and Analysis of Virtual Combinatorial Libraries Based on Defined Reaction Pathways; Book of Abstracts, p.P-29. Abstract Poster
  • Mordalski, S.; Kościółek, T.; Kristiansen, K.; Sylte, I.; Chilmonczyk, Z.; Bojarski, A.J.; A System for Automated Validation of GPCRs Homology Models Against Mutational Data; Book of Abstracts, p.P-45. Abstract Poster
  • Satała, G.; Duszyńska, B.; Nędza, K.; Bojarski, A.J.; Exploring the Effect of Radioligand Depletion on Affinity Determinations in the Dopamine D2 Binding Assay; Book of Abstracts, p.P-54. Abstract Poster
  • Smusz, S.; Kurczab, R. ; Bojarski, A.J.; Meta-Learning as an Improvement of Machine Learning Methods Performance in Virtual Screening; Book of Abstracts, p.P-57.Abstract Poster
  • Zajdel, P.; Marciniec, K.; Maślankiewicz, A.; Satała, G.; Wróbel, D.; Wesolowska, A.; Bojarski, A.J.; Pawłowski, M.; Synthesis and Pharmacological Evaluation of Quinolone- and Isoquinoline-Sulfonamides of Long-Chain Arylpiperazines as 5-HT7 Antagonists; Book of Abstracts, p.P-78. Abstract
  • Rataj, K.; Witek, J.; Kościółek, T.; Mordalski, S.; Bojarski, A.J.; Comparison of Homology Models of 5-HT6R Created with Different Crystal Templates; Book of Abstracts, p.P-52. Abstract Poster
  • Witek, J.; Rataj, K.; Kościółek, T.; Mordalski, S.; Bojarski, A.J.; Application of Interaction Patterns to Discriminate Ligand Preference to Target/Antitarget Protein; Book of Abstracts, p.P-73. Abstract Poster

10. 54th PTChem and SiTPChem Annual Meeting, 18-22.09.2011, Lublin, Poland

  • Zajdel, P.; Marciniec, K.; Piskorz, S.; Maślankiewicz, A.; Satała, G.; Partyka, A.; Jastrzębska-Więsek, M.; Wróbel, D.; Wesołowska, A.; Bojarski, A.J.; Pawłowski, M.; Chinolinosulfonamidy jako nowe ligandy receptorów 5-HT7; Book of Abstracts, p.389. Abstract

11. Schrödinger 11th Annual European User Group Meeting, 19-21.10.2011, Copenhagen, Denmark

  • Mordalski, S.; Kościółek, T.; Kristiansen, K.; Sylte, I.; Chilmonczyk, Z.; Bojarski, A.J.; A System for Automated Validation of GPCRs Homology Models Against Mutational Data; Book of Abstracts, p.15. Abstract

12.      7th International Meeting on Metabotropic Glutamate Receptors, 02-07.10.2011 Taormina, Italy

  • Brański, P.; Bojarski, A.; Burnat, G.; Chorobik, P.; Bugno, R.; Kurczab, R.; Staroń, J.; Chruścicka, B.; Pałucha-Poniewiara, A.; Pilc, A.; Searching for a new potential mGluR4 positive allosteric modulators; Curr. Neuropharmacol., 2011, 9, Suppl. 1.

13. 2nd Congress of Biochemistry and Cell Biology, 05-09.09.2011, Kraków, Poland

  • Walory, J.; Mielczarek, M.; Koronkiewicz, M.; Sylte, I. ; Bojarski, A.J.; Chilmonczyk, Z.; Cellular adenylate cyclase inhibition by the 6-nitroquipazine derivatives; Acta Biochim.Pol. 58, Suppl. 2, p.133.

14. Konferencja Naukowa Doktorantów Wydział Lekarskiego CMUJ, 11.05.2011, Kraków, Poland

  • Wróbel, D.; Partyka, A.; Jastrzębska-Więsek, M.; Zajdel, P.; Pawłowski, M.; Bojarski, A.J.; Satała, G.; Wesolowska, A.; Efekty funkcjonalne nowych sulfonoamidowych pochodnych 3-chinoliny w mysim modelu depresji;, Zeszyty Naukowe Towarzystwa Doktorantów UJ, 2011, 2, p.105.

15. V Kopernikańskie Seminarium Doktoranckie, 16-18.06.2011, Toruń, Poland

  • Wróbel, D.; Partyka, A.; Jastrzębska-Więsek, M.; Zajdel, P.; Pawłowski, M.; Bojarski, A.J.; Satała, G.; Wesolowska, A.; Efekty funkcjonalne nowych sulfonoamidowych ligandów receptora 5-HT7 w zwierzęcych modelach depresji u myszy; Book of Abstracts, p.86.