Conferences 2008

1. I Konwersatorium Chemii Medycznej, 19-20.09.2008, Lublin, Poland

  • Kościółek, T.; Dyduch, K. ; Szafrański, P.; Wróbel, T.; Nowak, M.; Homology Modelling as an Aid in Rational Synthesis of Nonclassical Cannabinoids; Book of Astracts, p.P-45. Abstract
  • Kurczab, R.; Nowak, M.; Bojarski, A.J.; Comparison of FlexX and Surflex Docking Algorithms Based on Astex Diverse Set; Book of Astracts, p.P-46. Abstract
  • Mordalski, S.; Lewgowd, W.; Stańczak, A.; Szczesio, M.; Główka, M.L.; Bojarski, A.J.; Experimental and Theoretical Studies on Conformations of Arylpiperazines with Pyrimido[5,4-c]quinolin-4(3H)-one Terminal; Book of Astracts, p.P-47. Abstract Poster

2. The Sixth Multidisciplinary Conference on Drug Research, 26-28.05.2008, Przemyśl, Poland

  • Jarończyk, M.; Chilmonczyk, Z.; Mazurek, A.P.; Nowak, G.; Bojarski, A.J.; Nowak, M.; Wołosewicz, K.; Sylte, I.; Kristiansen, K.; Ravna, A.W.; The ligand binding to the serotonin transporter; Book of Abstracts, p.6. Abstract
  • Duszyńska, B.; Bojarski, A.J.; Boksa, J.; Lenda, T.; Kamińska, D.; Cybulski, M.; Kaczmarek, Ł.S.; Searching for lead molecules as potential new CNS agents in the serotonin 5-HT6 screening assay; Book of Abstracts, p.23.Abstract Poster
  • Czopek, A.; Byrtus, H.; Kołaczkowski, M.; Wesołowska, A.; Bojarski, A.J.; Nędza, K.; Dybała, M.; Siwek, A.; Pawłowski, M.; Mannich base, 5-arylimidazolidine-2,4-dione derivatives with arylpiperazine moiety, as 5-HT1A receptor ligands with serotonin transporter affinity; Book of Abstracts , p.29. Abstract
  • Kowalski, P.; Kowalska, T.; Jaśkowska, J.; Butscher, M.; Duszyńska, B.; Flexible vs partly constrained linkers in NAN-190 and PK-13 analogs investigated as 5-HT1A/5-HT7 receptor ligands; Book of Abstracts, p.27.
  • Pieniążek, E.; Nowak, M.; Bojarski, A.J.; Jarończyk, M.; Chilmonczyk, Z.; Crystal structure of –adrenergic receptor as a new template in homology modeling of GPCR. Application to serotonin 5-HT1A and 5-HT7 receptors; Book of Abstracts, p.49. Abstract Poster
  • Herold, F.; Ciesielska, A.; Bojarski, A.J.; Nowak, G.; Synthesis of novel Pyrido[1,2-c]pyrimidine derivaives as selective ligands for 5-HT1A receptors; Book of Abstracts, p.28. Abstract
  • Żmudzki, P.; Chłoń-Rzepa, G.; Pawłowski, M.; Bojarski, A.J.; Duszyńska, B.; New serotonin receptors ligands in the group of 8-acylamide derivatives of 1,3-dimethyl-7-[(4-phenyl-piperazine-1-yl)-alkyl]-1H-purine-2,6-(3H,7H)-dione; Book of Abstracts, p.27. Abstract
  • Chłoń-Rzepa, G.; Żmudzki, P.; Pawłowski, M.; Bojarski, A.J.; Duszyńska, B.; Synthesis and serotonin receptor activity of new purine-2,6-dione derivatives with arylpiperazinylakloxyl moieties; Book of Abstracts, p.27.Abstract
  • Nowak, M.; Bojarski, A.J.; Salerno, L.; Modica, M.N.; Siracusa, M.A.; Molecular modeling explains differences in binding affinity of new potent and selective 5-HT1A ligands arylpiperazinylalkylthiobenzoxazole derivatives; Book of Abstracts, p.46. Abstract Poster
  • Paluchowska, M.H.; Nowak, M.; Synthesis and molecular modeling of 1,2,3,4-tetrahydroisoquinoline-based arylsulfonamides as potential 5-HT7 receptor ligandslines with imide fragment; Book of Abstracts, p.48. Abstract Poster
  • Paluchowska, M.H.; Kozioł, A.; Searching for the 5-HT7 receptor ligands in the series of new 1,2,3,4-tetrahydroisoquinolines with imide fragment; Book of Abstracts, p.48. Abstract Poster
  • Sikora, M.; Nowak, M.; Pharmacophore model of group II metabotrope glutamate receptor modulators; Book of Abstracts, p.46. Abstract
  • Zajdel, P.; Król, J.; Bojarski, A.J.; Duszyńska, B.; Scott, W.; Zhuo, Z.; O’Donnell, M.J.; Pawłowski, M.; Solid-phase synthesis and preliminary biological investigation of arylpiperazine library as 5-HT1A and 5-HT2A receptor ligands; Book of Abstracts, p.95.Abstract
  • Bugno, R.; Bojarski, A.J.; Nędza, K.; Kozioł, A.; 2-(1-Arylsulfonylpiperidin-2-yl)ethyl derivatives as 5-HT7 receptor ligands: sythesis and their affinity for 5-HT1A/5-HT2A/5-HT7/D2 receptors; Book of Abstracts, p.24. Abstract Poster
  • Bugno, R.; Bojarski, A.J.; Nędza, K.; Boksa, J.; SAR studies of novel 5-HT7R ligands with different spacers between aryl and amine moieties; Book of Abstracts, p.24. Abstract Poster
  • Nowak, M.; Mordalski, S.; Homology modelling of metabotropic glutamate receptor 2; Book of Abstracts, p.45.

3. BioInfo, 2008, Warszawa

  • Mordalski, S.; Butscher, M.; Bojarski, A.J.; Homology modelling of metabotropic glutamate receptor 3 extracellular domain.