Publications 1996

  1. Cegła, M. T.; Boksa, J.; Chojnacka-Wójcik, E.; Misztal, S. 4-Aryl-1-piperazinylalkyl derivatives of 1,2,3,4-tetrahydro-β-carboline ring system. Synthesis and preliminary in vivo studies. Pharmazie 1996, 51, 932-936 (http://www.ncbi.nlm.nih.gov/pubmed/8985983).
  2. Paluchowska, M. H.; Dereń-Wesołek, A.; Mokrosz, J. L.; Charakchieva-Minol, S.; Chojnacka-Wójcik, E. Analogs of MP 3022 with a Different Number of Nitrogen Atoms in the Heteroaromatic Fragment – New 5-HT1A Receptor Ligands . Arch. Pharm. (Weinheim) 1996, 32, 451-456 (http://www.ncbi.nlm.nih.gov/pubmed/8933747).
  3. Mokrosz, J. L.; Bojarski, A. J.; Harden, D. B.; Strekowski, L. Conformational Analysis of 4-(2‘-Furyl)-2-(methylamino)pyrimidine. J. Heterocyclic Chem. 1996, 33, 1207-1210 (http://onlinelibrary.wiley.com/doi/10.1002/jhet.5570330434/abstract).
  4. Mokrosz, J. L.; Duszyńska, B.; Charakchieva-Minol, S.; Bojarski, A. J.; Mokrosz, M. J.; Wydra, R. L.; Janda, L.; Strekowski, L. Structure-activity relationship studies of CNS agents. Part 29. N-Methylpiperazino-substituted derivatives of quinazoline, phthalazine and quinoline as novel α1, 5-HT 1A and 5-HT2A receptor ligands. Eur. J. Med. Chem. 1996, 31, 973-980 (http://scholar.qsensei.com/content/3wrsx).
  5. Byrtus, H.; Pawłowski, M.; Charakchieva-Minol, S.; Duszyńska, B.; Mokrosz, M. J.; Mokrosz, J. L.; Zejc, 3-(ω -Aminoalkyl)-5,5-dialkyl(or spirocycloalkyl-1,5-)hydantions as New 5-HT1A and 5-HT2A Receptor Ligands. Arch. Pharm. (Weinheim) 1996, 6, 283-290 (http://www.ncbi.nlm.nih.gov/pubmed/8767112).
  6. Mokrosz, J. L.; Dereń-Wesołek, A.; Tatarczyńska, E.; Duszyńska, B.; Bojarski, A. J.; Mokrosz, M. J.; Chojnacka-Wójcik, E. 8-{4-[2-(1,2,3,4-Tetrahydroisoquinolinyl)]-butyl}-9-azaspiro[4.5]decane-7,9-dione: A New 5-HT1A Receptor Ligand with the Same Activity Profile as Buspirone. J. Med. Chem. 1996, 39, 1125-1129 (http://www.ncbi.nlm.nih.gov/pubmed/8676348).
  7. Boksa, J.; Kłodzińska, A.; Charakchieva-Minol, S.; Chojnacka-Wójcik, E.; Mokrosz, J. L. Structure-activity relationship studies of CNS agents. Part 24. Analogs of N-tert-butyl-3-[4-(2-metoksyphenyl)-1-piperazinyl]-2-phenyl-propanamide (WAY – 100135). Pharmazie 1996, 51, 72-76 (http://www.ncbi.nlm.nih.gov/pubmed/8720802).